Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histone-lysine N-methyltransferase, H3 lysine-9 specific dim-5 (Neurospora crassa) | BDBM50315537 (CHEMBL1089316 | chaetocin) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Ludwig-Maximillians University of Munich Curated by ChEMBL | Assay Description Inhibition of Neurospora crassa DIM5 | Nat Chem Biol 1: 143-5 (2005) Article DOI: 10.1038/nchembio721 BindingDB Entry DOI: 10.7270/Q2PK0JZV | |||||||||||
More data for this Ligand-Target Pair |